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Dihexa vs PE 22-28

A side-by-side research comparison of Dihexa and PE 22-28 across mechanism, dosing, half-life, benefits, side effects and research status.

Comparison table

AttributeDihexaPE 22-28
Full nameDihexa (N-hexanoic-Tyr-Ile-(6)-aminohexanoic amide)PE 22-28 (Spadin-Derived TREK-1 Peptide)
CategoryCognitive & NootropicCognitive & Nootropic
StatusResearch compoundResearch peptide (preclinical)
MechanismAllosteric potentiator of HGF/c-Met signaling driving synaptogenesis, dendritic spine formation, and neuronal survival in hippocampal circuits.Selectively blocks the TREK-1 background potassium channel. TREK-1 inhibition enhances serotonergic signaling and rapidly increases synaptogenesis and neurogenesis, producing antidepressant-like effects faster than SSRIs in animal models.
Molecular weight507.6 Da~ (7-residue peptide)
Half-life6-12 hoursShort (peptide; improved vs spadin)
BioavailabilityModerate (oral/SubQ)Intranasal or injection (research)
Typical dose10-20 mg (oral) or 2-5 mg (SubQ)Not established for humans
FrequencyDailyResearch only
RouteOral or SubcutaneousIntranasal or injection (research)

Dihexa reported benefits

  • Dramatic synaptogenesis
  • Memory improvement
  • Cognitive restoration potential
  • Dendritic spine growth
  • HGF/c-Met activation

PE 22-28 reported benefits

  • Rapid antidepressant effects (preclinical)
  • Promotes neurogenesis and synaptogenesis
  • TREK-1 channel blockade
  • Neuroplasticity research interest

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Research and educational reference only. Not medical advice.