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5-Amino-1MQ vs Retatrutide

A side-by-side research comparison of 5-Amino-1MQ and Retatrutide across mechanism, dosing, half-life, benefits, side effects and research status.

Comparison table

Attribute5-Amino-1MQRetatrutide
Full name5-Amino-1-Methylquinolinium (NNMT Inhibitor)Retatrutide (Triple Agonist GIP/GLP-1/Glucagon)
CategoryWeight ManagementWeight Management
StatusResearch compoundPhase 3 Clinical Trial
MechanismInhibits NNMT enzyme, preventing methylation and degradation of nicotinamide. Increases intracellular NAD+ pools, activates sirtuins, and reduces fat cell size without affecting food intake.Triple agonism creates synergistic metabolic effects. Glucagon activation increases energy expenditure and hepatic fat oxidation while GLP-1/GIP reduce appetite and improve insulin sensitivity.
Molecular weight173.2 Da5,200 Da (approximate)
Half-life8-12 hours6 days
BioavailabilityHigh (oral)High (SubQ)
Typical dose50-100 mg1-2 mg → titrate up to 12 mg
Frequency1-2x dailyOnce weekly
RouteOral (capsule)Subcutaneous injection

5-Amino-1MQ reported benefits

  • Increased cellular energy metabolism
  • Reduced fat cell size
  • Elevated NAD+ levels
  • Does not suppress appetite
  • Improved muscle stem cell function
  • Oral convenience

Retatrutide reported benefits

  • Unprecedented weight loss (~24%)
  • Significant liver fat reduction
  • Improved cardiovascular markers
  • Enhanced energy expenditure
  • Superior glycemic control

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Research and educational reference only. Not medical advice.