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5-Amino-1MQ vs Tesofensine

A side-by-side research comparison of 5-Amino-1MQ and Tesofensine across mechanism, dosing, half-life, benefits, side effects and research status.

Comparison table

Attribute5-Amino-1MQTesofensine
Full name5-Amino-1-Methylquinolinium (NNMT Inhibitor)Tesofensine (Triple Monoamine Reuptake Inhibitor)
CategoryWeight ManagementWeight Management
StatusResearch compoundPhase 3 Clinical Trial
MechanismInhibits NNMT enzyme, preventing methylation and degradation of nicotinamide. Increases intracellular NAD+ pools, activates sirtuins, and reduces fat cell size without affecting food intake.Blocks presynaptic reuptake of noradrenaline, dopamine, and serotonin in the hypothalamus, enhancing satiety signaling, reducing food reward, and increasing thermogenesis.
Molecular weight173.2 Da329.4 Da
Half-life8-12 hours8-10 days
BioavailabilityHigh (oral)High (oral ~93%)
Typical dose50-100 mg0.25-0.5 mg
Frequency1-2x dailyOnce daily
RouteOral (capsule)Oral

5-Amino-1MQ reported benefits

  • Increased cellular energy metabolism
  • Reduced fat cell size
  • Elevated NAD+ levels
  • Does not suppress appetite
  • Improved muscle stem cell function
  • Oral convenience

Tesofensine reported benefits

  • Significant appetite reduction
  • Increased metabolic rate
  • Improved satiety signaling
  • 10-12% body weight loss
  • Oral administration convenience

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Research and educational reference only. Not medical advice.