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MOTS-c vs Tesofensine

A side-by-side research comparison of MOTS-c and Tesofensine across mechanism, dosing, half-life, benefits, side effects and research status.

Comparison table

AttributeMOTS-cTesofensine
Full nameMitochondrial Open Reading Frame of the 12S rRNA-cTesofensine (Triple Monoamine Reuptake Inhibitor)
CategoryWeight ManagementWeight Management
StatusResearch compoundPhase 3 Clinical Trial
MechanismActivates AMPK pathway, enhances mitochondrial metabolism, improves insulin sensitivity by increasing GLUT4 translocation, and promotes fatty acid oxidation.Blocks presynaptic reuptake of noradrenaline, dopamine, and serotonin in the hypothalamus, enhancing satiety signaling, reducing food reward, and increasing thermogenesis.
Molecular weight2,175 Da329.4 Da
Half-life4-8 hours8-10 days
BioavailabilityModerate (SubQ)High (oral ~93%)
Typical dose5-10 mg0.25-0.5 mg
Frequency3-5x per weekOnce daily
RouteSubcutaneous injectionOral

MOTS-c reported benefits

  • Exercise mimetic effects
  • Improved insulin sensitivity
  • Enhanced fat oxidation
  • Metabolic homeostasis
  • Anti-aging metabolic benefits
  • AMPK activation

Tesofensine reported benefits

  • Significant appetite reduction
  • Increased metabolic rate
  • Improved satiety signaling
  • 10-12% body weight loss
  • Oral administration convenience

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Research and educational reference only. Not medical advice.