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Noopept vs P21

A side-by-side research comparison of Noopept and P21 across mechanism, dosing, half-life, benefits, side effects and research status.

Comparison table

AttributeNoopeptP21
Full nameNoopept (GVS-111)P21 (CNTF-Derived Tetrapeptide)
CategoryCognitive & NootropicCognitive & Nootropic
StatusResearch compoundResearch compound
MechanismMetabolized to cycloprolylglycine which modulates AMPA/NMDA receptors. Increases NGF and BDNF in hippocampus/cortex. Antioxidant neuroprotection and acetylcholine enhancement.Mimics CNTF neurogenesis-enhancing portion by increasing BDNF and activating PI3K/Akt. Inhibits LIF signaling to selectively promote neural stem cell proliferation.
Molecular weight318.4 Da~450 Da
Half-life30-60 minutes (active metabolite longer)4-6 hours
BioavailabilityHigh (oral/sublingual)Moderate (crosses BBB)
Typical dose10-30 mg50-100 mcg/kg
Frequency2-3x dailyDaily
RouteOral or SublingualIntranasal or Subcutaneous

Noopept reported benefits

  • Enhanced memory/learning
  • Neuroprotection
  • BDNF/NGF increase
  • Improved focus
  • Anxiolytic
  • Low dose requirement

P21 reported benefits

  • Hippocampal neurogenesis
  • BDNF increase
  • Cognitive enhancement
  • BBB penetrant
  • No appetite suppression
  • Dendritic branching

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Research and educational reference only. Not medical advice.