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Pregnenolone vs Progesterone

A side-by-side research comparison of Pregnenolone and Progesterone across mechanism, dosing, half-life, benefits, side effects and research status.

Comparison table

AttributePregnenoloneProgesterone
Full namePregnenolone (Mother Hormone)Micronized Progesterone (Prometrium)
CategoryHormone ReplacementHormone Replacement
StatusOTC supplement / PrescribedFDA Approved
MechanismActs as the primary substrate for steroidogenesis (cortisol, DHEA, progesterone, testosterone, estrogen). Also functions as a neurosteroid, enhancing memory and NMDA receptor activity.Agonizes progesterone receptors and GABA-A receptors (via allopregnanolone metabolite). Inhibits 5-alpha reductase, opposes estrogen proliferative effects, and promotes myelination in neural tissue.
Molecular weight316.48 Da314.46 Da
Half-life~1-3 hours (oral)~16-18 hours (oral micronized)
Bioavailability~60% oral~10% oral (first-pass); ~100% topical/vaginal
Typical dose50-100 mg100-200 mg oral or 20-40 mg topical
FrequencyDaily (morning)Nightly (oral) or daily (topical)
RouteOral capsule or sublingualOral capsule, topical cream, or vaginal

Pregnenolone reported benefits

  • Hormone precursor balance
  • Memory enhancement
  • Mood improvement
  • Joint support
  • Myelin sheath repair
  • Stress resilience

Progesterone reported benefits

  • Enhanced deep sleep (GABA modulation)
  • Neuroprotection
  • Estrogen opposition
  • Reduced anxiety
  • DHT reduction (5AR inhibition)
  • Cardiovascular protection

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Research and educational reference only. Not medical advice.